Pharmacology

Biology / pharmacology.yaml
5 records
2 sections
pharmacokinetics 3 interactions 2

pharmacokinetics

DrugBioavailabilityHalf LifeProtein BindingMetabolismExcretion
Aspirin 50-68% 0.25h (parent), 3-6h (metabolite) 80-90% Liver (hydrolysis) Renal
Ibuprofen 80-100% 1.8-2h 90-99% Liver (CYP2C9) Renal
Metformin 50-60% 6.2h Negligible None Renal (unchanged)

interactions

Drug1Drug2MechanismSeverityDescription
Warfarin Aspirin Pharmacodynamic synergism (antiplatelet effect) Major Increased risk of bleeding.
Simvastatin Grapefruit Juice CYP3A4 inhibition Moderate Increased serum concentration of simvastatin.